Molecule Details
InChIKeyIKASAFLVQIJQOK-UVTDQMKNSA-N
Canonical SMILESCNS(=O)(=O)c1ccc(N/C=C2\C(=O)Nc3ccccc32)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.25
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB08122
Drug NameN-Methyl-4-{[(2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]amino}benzenesulfonamide
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: CHEMBL1234085 ChemSpider: 4450812 PDB: LS1 PubChem:5288708 PubChem:99444593 ZINC: ZINC000010254749
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 6.2 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.2 pIC50 TTD_MultiTarget
DrugBank Target Actions (1)
Target Gene Target Name Action Type
P24941 CDK2 Cyclin-dependent kinase 2 binder targets