Molecule Details
InChIKeyIJUYTPVJXNJDCI-UHFFFAOYSA-N
Canonical SMILESCc1cc(C)n2nc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CC(C)(C)CC5)CC4)cc3Oc3cc4cc[nH]c4c(F)c3F)nc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL10.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 10.4 Ki ChEMBL;BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 10.4 Ki ChEMBL;BindingDB