Molecule Details
InChIKeyIJTZHWGKWZMBCO-UHFFFAOYSA-N
Compound Name7-[4-[4-(8-hydroxy-2-oxochromen-5-yl)piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Canonical SMILESO=C1CCc2ccc(OCCCCN3CCN(c4ccc(O)c5oc(=O)ccc45)CC3)cc2N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB