Molecule Details
InChIKeyIIRIKFXWBJTDCC-UHFFFAOYSA-N
Compound Name4-[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]cyclohexane-1-carboxylic acid
Canonical SMILESO=C(O)C1CCC(N2CCN(C3=Cc4ccccc4Cn4ccnc43)CC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41595 HTR2B Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P35367 HRH1 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB