Molecule Details
InChIKeyIHTVZEPWUCPDDH-UHFFFAOYSA-N
Compound Name1-{1-[1-(Hydroxymethyl)cyclooctyl]piperidin-4-yl}-1Hbenzimidazol-2(3H)-one
Canonical SMILESO=c1[nH]c2ccccc2n1C1CCN(C2(CO)CCCCCCC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41146 OPRL1 Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB