Molecule Details
InChIKeyIHDRRZZOAOZYJS-UHFFFAOYSA-N
Compound Name2-(3,5-dimethylpiperazin-1-yl)-1-(1-(1-methylcyclooctyl)piperidin-4-yl)-1H-benzimidazole
Canonical SMILESCC1CN(c2nc3ccccc3n2C2CCN(C3(C)CCCCCCC3)CC2)CC(C)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41146 OPRL1 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB