Molecule Details
InChIKeyIGRIBIYYAXAWCQ-UHFFFAOYSA-N
Compound Name6-methyl-4-[3-[4-[2-(2,2,2-trifluoroethoxy)phenyl]piperazin-1-yl]propyl]-2H-1,2,4-triazine-3,5-dione
Canonical SMILESCc1n[nH]c(=O)n(CCCN2CCN(c3ccccc3OCC(F)(F)F)CC2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB