Molecule Details
InChIKeyIFMLEMDUMAPODC-XMMPIXPASA-N
Compound Name(3S)-3-(5-ethylthiophen-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
Canonical SMILESCCc1ccc([C@@H]2c3[nH]c4ccccc4c(=O)c3CN2c2ncc(-c3ccccn3)cn2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O76074 PDE5A Homo sapiens Human PF01590 PF00233 9.3 IC50 ChEMBL;BindingDB
P51160 PDE6C Homo sapiens Human PF01590 PF00233 8.9 IC50 ChEMBL;BindingDB
Q9HCR9 PDE11A Homo sapiens Human PF01590 PF00233 8.6 IC50 ChEMBL;BindingDB