Molecule Details
InChIKeyIFMIAYDNKIHTBR-XJAHMCCXSA-N
Compound Name3beta-(4-Methylphenyl)-2beta-[30-(4-chlorobenzyl)isoxazol-5-yl]-tropane hydrochloride
Canonical SMILESCc1ccc([C@H]2CC3CCC([C@H]2c2cc(Cc4ccc(Cl)cc4)no2)N3C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01959 SLC6A3 Homo sapiens Human PF00209 7.7 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.1 Ki ChEMBL;BindingDB
P23975 SLC6A2 Homo sapiens Human PF00209 6.1 Ki ChEMBL;BindingDB