Molecule Details
InChIKeyIFLPDVNBLNGRJS-UHFFFAOYSA-N
Compound Name6-(4-chlorophenyl)-2-(3,6-dihydro-2H-pyran-4-yl)-5-(1,5-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-5,6-dihydropyrrolo[3,4-d]imidazol-4(1H)-one
Canonical SMILESCc1cc(N2C(=O)c3nc(C4=CCOCC4)[nH]c3C2c2ccc(Cl)cc2)cn(C)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.5 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.4 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.1 IC50 ChEMBL;BindingDB