Molecule Details
InChIKeyIFEXCZMSTXWJSK-VQTJNVASSA-N
Compound Nametrans-(1R,2R)-2-pyridin-3-yl-N-[4-[3-(trifluoromethoxy)phenyl]sulfonylphenyl]cyclopropane-1-carboxamide
Canonical SMILESO=C(Nc1ccc(S(=O)(=O)c2cccc(OC(F)(F)F)c2)cc1)[C@@H]1C[C@H]1c1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43490 NAMPT Homo sapiens Human PF18127 PF04095 8.0 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.6 IC50 ChEMBL
P11712 CYP2C9 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB