Molecule Details
InChIKeyIENQHTKISQTRDU-XGTKUTNFSA-N
Compound NameN-[(4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]-2-cyanopyridine-4-carboxamide
Canonical SMILESN#Cc1cc(C(=O)N[C@@H]2CC[C@@]3(O)[C@H]4Cc5ccc(O)c6c5[C@@]3(CCN4CC3CC3)[C@H]2O6)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.9 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB