Molecule Details
InChIKeyIEHBGAHJQRMSCS-VABKMULXSA-N
Compound Name(2S,5S,8S)-2-butyl-5-[4-(ethanethioylamino)butyl]-3,6,14,21-tetraoxo-1,4,7,13-tetrazacyclohenicosane-8-carboxamide
Canonical SMILESCCCC[C@@H]1NC(=O)CCCCCCC(=O)NCCCC[C@@H](C(N)=O)NC(=O)[C@H](CCCCNC(C)=S)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96EB6 SIRT1 Homo sapiens Human PF02146 6.7 IC50 ChEMBL;BindingDB
Q8IXJ6 SIRT2 Homo sapiens Human PF02146 6.6 IC50 ChEMBL;BindingDB
Q9NTG7 SIRT3 Homo sapiens Human PF02146 6.3 IC50 ChEMBL;BindingDB