Molecule Details
InChIKeyIDAHTGCAQFARTJ-UHFFFAOYSA-N
Compound Name2-[4-[1-[6-(1,4-Diazepan-1-yl)-2-pyridinyl]pyrazolo[4,3-c]pyridin-6-yl]pyrazol-1-yl]acetamide
Canonical SMILESNC(=O)Cn1cc(-c2cc3c(cn2)cnn3-c2cccc(N3CCCNCC3)n2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.7 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.6 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB