Molecule Details
InChIKeyICYGLDQWNJHCEE-UHFFFAOYSA-N
Compound NameN-[5-[(3,5-difluorophenyl)methyl]-1H-indazol-3-yl]-2-(2-methoxyethylamino)-4-(4-methylpiperazin-1-yl)benzamide
Canonical SMILESCOCCNc1cc(N2CCN(C)CC2)ccc1C(=O)Nc1n[nH]c2ccc(Cc3cc(F)cc(F)c3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UM73 ALK Homo sapiens Human PF12810 PF00629 PF07714 6.4 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.2 IC50 ChEMBL
Q96GD4 AURKB Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB