Molecule Details
InChIKeyICVMJXJRTYOTJH-UHFFFAOYSA-N
Compound Name(2-{[2-(2-Sulfamoyl-benzothiazol-6-yloxy)-ethoxycarbonylmethyl]-amino}-ethylamino)-acetic acid
Canonical SMILESNS(=O)(=O)c1nc2ccc(OCCOC(=O)CNCCNCC(=O)O)cc2s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.06
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.4 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.4 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.4 Ki ChEMBL;BindingDB