Molecule Details
InChIKeyICODOOXDNPOINQ-UHFFFAOYSA-N
Compound Name4-[3-[[[4-(Trifluoromethyl)benzoyl]amino]methyl]anilino]quinazoline-8-carboxamide
Canonical SMILESNC(=O)c1cccc2c(Nc3cccc(CNC(=O)c4ccc(C(F)(F)F)cc4)c3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.8 IC50 ChEMBL;BindingDB