Molecule Details
InChIKeyIBQHDBZMXPNKAU-UHFFFAOYSA-N
Compound NameN-(3-fluorophenyl)-2-(2-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-1,3-thiazol-5-yl)acetamide
Canonical SMILESCOCCOc1cc2ncnc(Nc3ncc(CC(=O)Nc4cccc(F)c4)s3)c2cc1OC
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 9.0 pIC50 TTD_MultiTarget