Molecule Details
InChIKeyIBAUSYCHSXHDOA-UHFFFAOYSA-N
Compound Name4-[(4-Anilino-5-fluoropyrimidin-2-yl)amino]benzamide
Canonical SMILESNC(=O)c1ccc(Nc2ncc(F)c(Nc3ccccc3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.8
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.3 IC50 ChEMBL
Q96GD4 AURKB Homo sapiens Human PF00069 7.8 IC50 ChEMBL
O60674 JAK2 Homo sapiens Human PF18379 PF18377 PF17887 PF07714 PF21990 7.3 IC50 ChEMBL