Molecule Details
InChIKeyIAUGVDTWTMEFGP-UHFFFAOYSA-N
Compound Name2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2,6-dimethyl-1Hindol-4-yloxy)acetic acid
Canonical SMILESCc1cc(OCC(=O)O)c2c(C(=O)C(N)=O)c(C)n(Cc3ccccc3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NZK7 PLA2G2E Homo sapiens Human PF00068 6.9 IC50 ChEMBL;BindingDB
P14555 PLA2G2A Homo sapiens Human PF00068 6.5 IC50 ChEMBL;BindingDB
P39877 PLA2G5 Homo sapiens Human PF00068 6.1 IC50 ChEMBL;BindingDB