Molecule Details
InChIKeyIAOOIOSKSIPSBX-UHFFFAOYSA-N
Compound Name2-[[4-Hydroxy-1-[[4-(2-hydroxypropan-2-yl)phenyl]methyl]-2-oxo-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
Canonical SMILESCC(C)(O)c1ccc(Cn2c3c(c(O)c(C(=O)NCC(=O)O)c2=O)COC3)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96KS0 EGLN2 Homo sapiens Human PF13640 8.2 IC50 ChEMBL;BindingDB
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 8.2 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 7.8 IC50 ChEMBL;BindingDB