Molecule Details
InChIKeyHZTZFAQVGYSTHZ-UHFFFAOYSA-N
Compound Name2-[2-(cyclobutanecarbonylamino)-4-pyridinyl]-4-(cyclopropylmethoxy)-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-1,3-thiazole-5-carboxamide
Canonical SMILESO=C(NCCCNc1c2c(nc3ccccc13)CCCC2)c1sc(-c2ccnc(NC(=O)C3CCC3)c2)nc1OCC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06276 BCHE Homo sapiens Human PF08674 PF00135 7.5 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P22303 ACHE Homo sapiens Human PF08674 PF00135 6.5 IC50 ChEMBL;BindingDB