Molecule Details
InChIKeyHZPJCVFFDAMKRH-UHFFFAOYSA-N
Compound Name3-(8-methylimidazo[1,2-a] pyridin-3-yl)-2-(1H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESCc1cccn2c(-c3cccc(S(N)(=O)=O)c3-c3nnn[nH]3)cnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.15
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.2 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 8.2 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 7.0 IC50 BindingDB