Molecule Details
InChIKeyHYUPCNJXAHVNMI-CVEARBPZSA-N
Compound Name2-(((S)-1-((R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl)pyrrolidin-2-yl)methylamino)nicotinonitrile
Canonical SMILESN#Cc1cccnc1NC[C@@H]1CCCN1C(=O)C[C@H](N)Cc1cc(F)c(F)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 8.5 IC50 ChEMBL;BindingDB
P10635 CYP2D6 Homo sapiens Human PF00067 6.2 IC50 ChEMBL;BindingDB
Q9UHL4 DPP7 Homo sapiens Human PF05577 6.2 IC50 ChEMBL;BindingDB