Molecule Details
InChIKeyHYBCPKCAHCAFSQ-UHFFFAOYSA-N
Compound NameN-(2-(dimethylamino)ethyl)-4-((4-(imidazo(1,2-a)pyridin-3-yl)pyrimidin-2-yl)amino)benzene-1-sulfonamide
Canonical SMILESCN(C)CCN[S@SP3](=O)(=O)c1ccc(Nc2nccc(-c3cnc4ccccn34)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.14
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 8.3 pIC50 TTD_MultiTarget
P06493 CDK1 Homo sapiens Human PF00069 8.1 pIC50 TTD_MultiTarget
P11802 CDK4 Homo sapiens Human PF00069 8.1 pIC50 TTD_MultiTarget