Molecule Details
InChIKeyHXWCQEQIPYCSAM-QPPBQGQZSA-N
Compound Name2-((3,4-dichlorophenyl)(methyl)amino)-1-((2R,3R)-3-phenyl-2-(pyrrolidin-1-ylmethyl)piperidin-1-yl)ethanone
Canonical SMILESCN(CC(=O)N1CCC[C@H](c2ccccc2)[C@@H]1CN1CCCC1)c1ccc(Cl)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UKP6 UTS2R Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P10635 CYP2D6 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB