Molecule Details
InChIKeyHXQNEKJQBGXFAG-UHFFFAOYSA-N
Compound Name(Rac)-AMG8379
Canonical SMILESCOc1cc(-c2cc(F)cc(Cl)c2)c(F)cc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ccon3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01118 SCN7A Homo sapiens Human PF00520 PF24609 PF06512 8.5 IC50 ChEMBL;BindingDB
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 8.1 IC50 ChEMBL;BindingDB