Molecule Details
InChIKeyHXPQWNPLNIEJOW-UHFFFAOYSA-N
Compound Name2-(4-((2-Ethyl-5,7-dimethylpyrazolo(1,5-a)pyrimidin-3-yl)methyl)phenyl)-5-(piperidin-4-yl)-1,3,4-oxadiazole
Canonical SMILESCCc1nn2c(C)cc(C)nc2c1Cc1ccc(-c2nnc(C3CCNCC3)o2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P46093 GPR4 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
P46098 HTR3A Homo sapiens Human PF02931 PF02932 6.4 Ki ChEMBL
Q5BJF2 TMEM97 Homo sapiens Human PF05241 6.3 Ki ChEMBL