Molecule Details
InChIKeyHXPLFONFARJCJA-UHFFFAOYSA-N
Compound Name4-fluoro-N-[3-[1-[7-[4-[5-[(4-fluorobenzoyl)amino]-1H-indol-3-yl]piperidin-1-yl]heptyl]piperidin-4-yl]-1H-indol-5-yl]benzamide
Canonical SMILESO=C(Nc1ccc2[nH]cc(C3CCN(CCCCCCCN4CCC(c5c[nH]c6ccc(NC(=O)c7ccc(F)cc7)cc56)CC4)CC3)c2c1)c1ccc(F)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.2 IC50 ChEMBL;BindingDB