Molecule Details
InChIKeyHXHKXXRIQOWOHI-UHFFFAOYSA-N
Compound Name8-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-amine
Canonical SMILESCOc1cc2c(cc1OC)CN(Cc1cnc(N)n3nc(-c4ccco4)nc13)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB