Molecule Details
InChIKeyHXHFVYQPJRIKLE-DLBZAZTESA-N
Compound Name(3R,5S)-5-amino-1-[3-[[2-(2,6-difluorophenyl)quinolin-8-yl]amino]-4-pyridinyl]piperidin-3-ol
Canonical SMILESN[C@H]1C[C@@H](O)CN(c2ccncc2Nc2cccc3ccc(-c4c(F)cccc4F)nc23)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB