Molecule Details
InChIKeyHXENBKGGEPBXOQ-UHFFFAOYSA-N
Compound NameUS9890166, Example 54
Canonical SMILESCOc1ncc(-c2nc3c(n2C)C(c2ccc(Cl)cc2)N(c2cc(OC)c4nnc(C)n4c2)C3=O)c(OC)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.2 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.0 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 6.9 IC50 ChEMBL;BindingDB