Molecule Details
InChIKeyHWZRSTGNKARGTN-UHFFFAOYSA-N
Compound Name4-[4-chloro-2-(1H-pyrazol-5-yl)phenoxy]-3-cyano-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
Canonical SMILESN#Cc1cc(S(=O)(=O)Nc2ncns2)ccc1Oc1ccc(Cl)cc1-c1ccn[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.5 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 6.7 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.4 IC50 ChEMBL;BindingDB