Molecule Details
InChIKeyHWYWVGSBHACYHO-UHFFFAOYSA-N
Compound Name1-[4-(6-Bromo-13-chloro-17-methyl-4,15-diazatetracyclo[9.7.0.03,8.014,18]octadeca-1(18),3(8),4,6,11,13,16-heptaen-2-ylidene)piperidin-1-yl]-2-(1-oxidopyridin-1-ium-4-yl)ethanone
Canonical SMILESCc1c[nH]c2c(Cl)cc3c(c12)C(=C1CCN(C(=O)Cc2cc[n+]([O-])cc2)CC1)c1ncc(Br)cc1CC3
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.24
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.2 IC50 ChEMBL;BindingDB