Molecule Details
InChIKeyHWKYDSTYDOMPPO-UHFFFAOYSA-N
Compound Name1-[2-[[1-(4-Bromophenyl)-5-(4-methylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-hydroxyurea
Canonical SMILESCS(=O)(=O)c1ccc(-c2nc(SCCN(O)C(N)=O)nn2-c2ccc(Br)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35354 PTGS2 Homo sapiens Human PF03098 6.8 IC50 ChEMBL;BindingDB
P09917 ALOX5 Homo sapiens Human PF00305 PF01477 6.1 IC50 ChEMBL;BindingDB