Molecule Details
InChIKeyHWAQNGBXVSEQHM-UHFFFAOYSA-N
Compound Name5-(5-methyl-3-pyridinyl)-3-(6-piperazin-1-yl-2-pyridinyl)-1H-pyrazolo[3,4-c]pyridine
Canonical SMILESCc1cncc(-c2cc3c(-c4cccc(N5CCNCC5)n4)n[nH]c3cn2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.4 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 10.4 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB