Molecule Details
InChIKeyHVSUPPZVIPTMEM-UHFFFAOYSA-N
Compound Name7-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one
Canonical SMILESCOc1ccccc1N1CCN(CCCCOc2ccc3c(c2)NC(=O)CC3)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB