Molecule Details
InChIKeyHVRRMJKBJSKZOK-UHFFFAOYSA-N
Compound NamePyrazolo[4,3-h]quinazoline-3-carboxamide, 36
Canonical SMILESCNC(=O)c1nn(C)c2c1C(C)(C)Cc1cnc(Nc3ccc(CN4CCOCC4)cc3)nc1-2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.86
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.4 pIC50 TTD_MultiTarget
O14965 AURKA Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB