Molecule Details
InChIKeyHVRASXRMCOQSPI-UHFFFAOYSA-N
Compound NameN-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-5-[4-(2-methylphenyl)phenyl]-1,3,4-oxadiazol-2-amine
Canonical SMILESCc1ccccc1-c1ccc(-c2nnc(N(C)Cc3ccc4nccn4c3)o2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12866 MERTK Homo sapiens Human PF00041 PF00047 PF13927 PF07714 7.9 IC50 ChEMBL;BindingDB
P30530 AXL Homo sapiens Human PF00041 PF13927 PF07714 6.2 IC50 ChEMBL;BindingDB
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.0 IC50 ChEMBL;BindingDB