Molecule Details
InChIKeyHVNQYDHDQBJAAH-ZDUSSCGKSA-N
Compound Nametert-butyl N-[(3S)-1-[2-amino-6-(3-amino-1H-indazol-6-yl)pyrimidin-4-yl]piperidin-3-yl]carbamate
Canonical SMILESCC(C)(C)OC(=O)N[C@H]1CCCN(c2cc(-c3ccc4c(N)n[nH]c4c3)nc(N)n2)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.33
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 6.5 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 6.0 IC50 ChEMBL;BindingDB