Molecule Details
InChIKeyHVNQYDHDQBJAAH-CYBMUJFWSA-N
Compound Name1,1-Dimethylethyl {(3R)-1-[2-amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-3-piperidinyl}carbamate
Canonical SMILESCC(C)(C)OC(=O)N[C@@H]1CCCN(c2cc(-c3ccc4c(N)n[nH]c4c3)nc(N)n2)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 7.6 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 Clinical TTD_MultiTarget TTD_MultiTarget