Molecule Details
InChIKeyHVLBTSWQHJSANX-UHFFFAOYSA-N
Compound Name4-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-benzoic acid
Canonical SMILESO=C(O)c1ccc(-c2[nH]nc3cc(Nc4ccccc4Cl)ccc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB