Molecule Details
InChIKeyHVKVREKLPAMYHA-IBGZPJMESA-N
Compound Name5-cyclopropyl-2-(3,5-dimethoxyanilino)-7-[[(2S)-1-hydroxy-3-phenylpropan-2-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carboxamide
Canonical SMILESCOc1cc(Nc2nn3c(N[C@H](CO)Cc4ccccc4)cc(C4CC4)nc3c2C(N)=O)cc(OC)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 8.2 IC50 ChEMBL;BindingDB
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 7.8 IC50 ChEMBL;BindingDB