Molecule Details
InChIKeyHVHBXBDAWFYVOJ-UHFFFAOYSA-N
Compound NameN2-methyl-N4-(5-methyl-1H-pyrazol-3-yl)-N2-phenylquinazoline-2,4-diamine
Canonical SMILESCc1cc(Nc2nc(N(C)c3ccccc3)nc3ccccc23)n[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 6.5 Ki ChEMBL;BindingDB