Molecule Details
InChIKeyHVFIZGFUTYQRCG-UHFFFAOYSA-N
Compound NameN-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-4-(trifluoromethyl)-1,2,7,8-tetrahydrofuro[3,2-e]indole-6-carboxamide
Canonical SMILESCc1ncccc1Oc1ccc(NC(=O)N2CCc3c2cc(C(F)(F)F)c2c3CCO2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB