Molecule Details
InChIKeyHUPNMGIBODMDOH-UHFFFAOYSA-N
Compound NameN-(5-(3-chloropyridin-4-yl)-6-(pyridin-2-yl)pyrazin-2-yl)cyclopropanecarboxamide
Canonical SMILESO=C(Nc1cnc(-c2ccncc2F)c(-c2ccncc2)n1)C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P33261 CYP2C19 Homo sapiens Human PF00067 6.2 Ki ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.0 IC50 ChEMBL;BindingDB