Molecule Details
InChIKeyHUJUWOZUJZKBDW-UHFFFAOYSA-N
Compound Name1-Methyl-5-[3-methyl-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-1,4,5,10-tetrahydropyrazolo[3,4-b][1,5]benzodiazepine
Canonical SMILESCc1ccn(-c2ccc(C(=O)N3Cc4cnn(C)c4Nc4ccccc43)cc2C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 7.7 Ki ChEMBL;BindingDB
P30559 OXTR Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P30518 AVPR2 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB