Molecule Details
InChIKeyHTYIYAXOMLBJLR-HSZRJFAPSA-N
Canonical SMILESCCc1[nH]c2nc1-c1ccc(NC(=O)OC)cc1NC(=O)CCCC[C@@H]2c1ccc(-c2c(F)cccc2-n2cc(C(F)(F)F)cn2)c[n+]1[O-]
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 8.6 Ki ChEMBL;BindingDB
P06870 KLK1 Homo sapiens Human PF00089 6.2 Ki ChEMBL;BindingDB