Molecule Details
InChIKeyHTRVDWTYRAEJCW-UHFFFAOYSA-N
Compound Name4-[3-(5-Aminomethyl-thiazol-2-ylamino)-benzylamino]-quinazoline-8-carboxylic acid amide
Canonical SMILESNCc1cnc(Nc2cccc(CNc3ncnc4c(C(N)=O)cccc34)c2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.7 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 9.1 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.0 IC50 ChEMBL;BindingDB