Molecule Details
InChIKeyHTCXYVHODSQMOP-UHFFFAOYSA-N
Compound Name3-[(7-Chloro-2-oxo-2H-chromen-4-ylmethyl)-amino]-N-(5-sulfamoyl-[1,3,4]thiadiazol-2-yl)-propionamide
Canonical SMILESNS(=O)(=O)c1nnc(NC(=O)CCNCc2cc(=O)oc3cc(Cl)ccc23)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.44
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.7 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB